Aminoacids with a contribution to the binding affinity, but with low correlation to experimental deltaG values --> PLS coefficients near zero.
Interactions, which are important for general ligand binding and do not vary among the given receptor-ligand complexes of a training set, have a low correlation to the experimental binding affinity and their PLS coefficients is near zero.

|mean (energy terms)| >= 0.01 and standard deviation (energy terms) <= 0.01 and |PLS coefficient| <= 0.001


thrombin (E)
trypsin (B)
urokinase (A)
vdW
T139
S139


G140
G140


V158

T158


A160




I163

G184



Y184A




L185
D185


G187


G188
G188



K188A




P198

F199
V199



K222



N223

elec


I17



Y40

V158

T158


A160



L163


G184




G188



G197




P198

F199

L199


T229
T229

C:\Daten\COMBINE_paper\work121006\
A_urokinase_active-nodbl-A25-A28-A29.dat.table.transpose.xls
B_trypsin_active-nodbl-A98-B07-A96-A04-B17.dat.table.transpose.xls
E_thrombin_output-A12_1-A09-A84-A88-A89-A90.dat.table.transpose.xls


SH 15.03.2007
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